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Anti Malarials APIs

Artemisinin derivatives, quinoline alkaloids, and cinchona-based APIs for ACT and parenteral malaria regimens. Supplied in USP/EP/BP grade to manufacturers serving endemic and non-endemic export markets.

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All Anti Malarials APIs

12 APIs available

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CAS 75887-54-6 Product Code AM-001 WHO-GMP

Alpha Beta Arteether

Semi-synthetic artemisinin derivative in USP-aligned grade, traded as an oily solution for IM injectable manufacturing. Sourced for severe and cerebral malaria treatment, typically in 30:70 alpha:beta isomer ratio.

USP Injection
Anti Malarials API

Alpha Beta Arteether

CAS
75887-54-6
Product Code
AM-001
Category
Anti Malarials
Specification
USP
Quality
WHO-GMP
Applications
Injection

Full description

Semi-synthetic artemisinin derivative in USP-aligned grade, traded as an oily solution for IM injectable manufacturing. Sourced for severe and cerebral malaria treatment, typically in 30:70 alpha:beta isomer ratio.

CAS 86-42-0 / 69-44-3 Product Code AM-002 WHO-GMP

Amodiaquine Base / HCl

4-aminoquinoline antimalarial supplied as free base (86-42-0) and hydrochloride salt (69-44-3) — USP/EP/BP grade — for oral tablet and suspension manufacturing. Sourced for ACT combination with artesunate against P. falciparum and P. vivax.

USP EP BP Oral
Anti Malarials API

Amodiaquine Base / HCl

CAS
86-42-0 / 69-44-3
Product Code
AM-002
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral

Full description

4-aminoquinoline antimalarial supplied as free base (86-42-0) and hydrochloride salt (69-44-3) — USP/EP/BP grade — for oral tablet and suspension manufacturing. Sourced for ACT combination with artesunate against P. falciparum and P. vivax.

CAS 71963-77-4 Product Code AM-003 WHO-GMP

Artemether

Methyl ether derivative of artemisinin in USP/EP/BP/JP grade for oral and injectable formulation manufacturing. Core API in artemether-lumefantrine fixed-dose ACT for multi-drug-resistant P. falciparum.

USP EP BP JP Oral Injection
Anti Malarials API

Artemether

CAS
71963-77-4
Product Code
AM-003
Category
Anti Malarials
Specification
USP / EP / BP / JP
Quality
WHO-GMP
Applications
Oral · Injection

Full description

Methyl ether derivative of artemisinin in USP/EP/BP/JP grade for oral and injectable formulation manufacturing. Core API in artemether-lumefantrine fixed-dose ACT for multi-drug-resistant P. falciparum.

CAS 88495-63-0 Product Code AM-004 WHO-GMP

Artesunate Plain / Sterile

Water-soluble artemisinin derivative traded in plain grade for oral/rectal formulations and sterile grade (USP <797> processed) for IV/IM injectable manufacturing. Same active compound across both grades — used for severe and uncomplicated malaria.

USP Oral Injection Rectal
Anti Malarials API

Artesunate Plain / Sterile

CAS
88495-63-0
Product Code
AM-004
Category
Anti Malarials
Specification
USP
Quality
WHO-GMP
Applications
Oral · Injection · Rectal

Full description

Water-soluble artemisinin derivative traded in plain grade for oral/rectal formulations and sterile grade (USP <797> processed) for IV/IM injectable manufacturing. Same active compound across both grades — used for severe and uncomplicated malaria.

CAS 50-63-5 Product Code AM-005 WHO-GMP

Chloroquine Phosphate

Classic 4-aminoquinoline antimalarial in USP/EP/BP grade for oral tablet manufacturing. Sourced for prophylaxis and treatment of chloroquine-susceptible P. vivax and P. falciparum strains.

USP EP BP Oral
Anti Malarials API

Chloroquine Phosphate

CAS
50-63-5
Product Code
AM-005
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral

Full description

Classic 4-aminoquinoline antimalarial in USP/EP/BP grade for oral tablet manufacturing. Sourced for prophylaxis and treatment of chloroquine-susceptible P. vivax and P. falciparum strains.

CAS 71939-50-9 Product Code AM-006 WHO-GMP

Dihydro Artemisinin

Active artemisinin metabolite in USP/EP grade for oral tablet and capsule formulation manufacturing. Supplied both as the reduction intermediate behind artemether/artesunate metabolism and for standalone ACT formulations.

USP EP Oral
Anti Malarials API

Dihydro Artemisinin

CAS
71939-50-9
Product Code
AM-006
Category
Anti Malarials
Specification
USP / EP
Quality
WHO-GMP
Applications
Oral

Full description

Active artemisinin metabolite in USP/EP grade for oral tablet and capsule formulation manufacturing. Supplied both as the reduction intermediate behind artemether/artesunate metabolism and for standalone ACT formulations.

CAS 82186-77-4 Product Code AM-007 WHO-GMP

Lumefantrine

Aryl amino alcohol antimalarial in USP/EP/BP/IP grade for fixed-dose combination tablet manufacturing alongside artemether. Core partner compound in WHO-recommended ACT regimens for P. falciparum.

USP EP BP IP Oral
Anti Malarials API

Lumefantrine

CAS
82186-77-4
Product Code
AM-007
Category
Anti Malarials
Specification
USP / EP / BP / IP
Quality
WHO-GMP
Applications
Oral

Full description

Aryl amino alcohol antimalarial in USP/EP/BP/IP grade for fixed-dose combination tablet manufacturing alongside artemether. Core partner compound in WHO-recommended ACT regimens for P. falciparum.

CAS 51773-92-3 Product Code AM-008 WHO-GMP

Mefloquine

Quinolinemethanol antimalarial supplied as hydrochloride salt — USP grade — for oral tablet manufacturing. Sourced for prophylaxis and treatment of multi-drug-resistant P. falciparum malaria.

USP Oral
Anti Malarials API

Mefloquine

CAS
51773-92-3
Product Code
AM-008
Category
Anti Malarials
Specification
USP
Quality
WHO-GMP
Applications
Oral

Full description

Quinolinemethanol antimalarial supplied as hydrochloride salt — USP grade — for oral tablet manufacturing. Sourced for prophylaxis and treatment of multi-drug-resistant P. falciparum malaria.

CAS 63-45-6 Product Code AM-009 WHO-GMP

Primaquine Phosphate

8-aminoquinoline radical curative agent in USP/EP/BP grade for oral tablet manufacturing. Sourced for hepatic hypnozoite elimination in P. vivax and P. ovale relapse prevention.

USP EP BP Oral
Anti Malarials API

Primaquine Phosphate

CAS
63-45-6
Product Code
AM-009
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral

Full description

8-aminoquinoline radical curative agent in USP/EP/BP grade for oral tablet manufacturing. Sourced for hepatic hypnozoite elimination in P. vivax and P. ovale relapse prevention.

CAS 60-93-5 Product Code AM-010 WHO-GMP

Quinine Di Hydrochloride

Water-soluble cinchona alkaloid salt in USP/EP/BP grade for injectable solution manufacturing. Sourced for parenteral treatment of severe malaria where oral administration is not feasible.

USP EP BP Oral Injection
Anti Malarials API

Quinine Di Hydrochloride

CAS
60-93-5
Product Code
AM-010
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral · Injection

Full description

Water-soluble cinchona alkaloid salt in USP/EP/BP grade for injectable solution manufacturing. Sourced for parenteral treatment of severe malaria where oral administration is not feasible.

CAS 6119-47-7 Product Code AM-011 WHO-GMP

Quinine Hydrochloride

Cinchona alkaloid hydrochloride dihydrate in USP/EP/BP grade for injectable and oral formulation manufacturing. Supplied for severe malaria protocols requiring parenteral or oral alkaloid therapy.

USP EP BP Oral Injection
Anti Malarials API

Quinine Hydrochloride

CAS
6119-47-7
Product Code
AM-011
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral · Injection

Full description

Cinchona alkaloid hydrochloride dihydrate in USP/EP/BP grade for injectable and oral formulation manufacturing. Supplied for severe malaria protocols requiring parenteral or oral alkaloid therapy.

CAS 549-56-4 Product Code AM-012 WHO-GMP

Quinine Sulphate

Cinchona bark-derived alkaloid sulfate salt in USP/EP/BP grade for oral tablet and suspension manufacturing. Sourced for uncomplicated and severe malaria treatment in combination regimens.

USP EP BP Oral
Anti Malarials API

Quinine Sulphate

CAS
549-56-4
Product Code
AM-012
Category
Anti Malarials
Specification
USP / EP / BP
Quality
WHO-GMP
Applications
Oral

Full description

Cinchona bark-derived alkaloid sulfate salt in USP/EP/BP grade for oral tablet and suspension manufacturing. Sourced for uncomplicated and severe malaria treatment in combination regimens.

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